論文・特許

事業を通して得られた知見や成果を社会に還元するため、学会発表、論文投稿、特許取得を行っています。

■最近の投稿論文・総説

Development of Hamari Ligands for Practical Asymmetric Synthesis of Tailor-Made 続きを読む...
Practical Method for Preparation of (S)-2-Amino-5,5,5-trifluoropentanoic Acid vi 続きを読む...
Large‐Scale Asymmetric Synthesis of Fmoc‐(S)‐2‐Amino‐6,6,6‐Trifluorohexanoic Aci 続きを読む...
Optical Resolution of Rimantadine. Molecules 2019, 24, 1828. DOI: 10.3390/molecu 続きを読む...
Convenient Asymmetric Synthesis of Fmoc-(S)-6,6,6-Trifluoro-Norleucine. Symmetry 続きを読む...
Expedient Asymmetric Synthesis of (S)‑2-Amino-4,4,4-trifluorobutanoic Acid via A 続きを読む...
Large Scale Synthesis of Chiral (3Z,5Z)‑2,7-Dihydro‑1H‑azepine-Derived Hamari Li 続きを読む...
Tandem alkylation−second-order asymmetric transformation protocol for the prepar 続きを読む...
Second-order asymmetric transformation and its application for the practical syn 続きを読む...
2-Pyrrolidinecarboxamide, N-(2-Benzoyl-4-chlorophenyl)-1-[(3,4-dichlorophenyl)me 続きを読む...

■特許

  1. METHOD FOR SYNTHESIZING OPTICALLY ACTIVE α-AMINO ACID USING CHIRAL METAL COMPLEX COMPRISING AXIALLY CHIRAL N-(2-ACYLARYL)-2-[5,7-DIHYDRO-6H-DIBENZO[c,e]AZEPIN-6-YL]ACETAMIDE COMPOUND AND AMINO ACID. WO2014188783.
  2. AXIAL-ASYMMETRIC N-(2-ACYLARYL)-2-[5, 7-DIHYDRO-6H-DIBENZO [C, E] AZEPINE-6-YL] ACETAMIDE COMPOUND AND CHIRALITY CONVERSION METHOD FOR [Alpha]-AMINO ACID USING SAME. WO2014098063.
  3. METHOD FOR PRODUCING OPTICALLY ACTIVE ALCOHOL. WO2013061999.
  4. METHOD FOR PRODUCING OPTICALLY ACTIVE TETRAHYDROQUINOLINE. WO2013011930.
  5. METHOD FOR PRODUCING FINE POWDER OF LOXOPROFEN SODIUM DIHYDRATE FOR PHARMACEUTICAL PREPARATIONS. WO2012137667.
  6. NOVEL DIHYDROTRIAZINE DERIVATIVE. WO2010024225.
  7. PROCESS FOR PRODUCTION OF ETHYNYLTHYMIDINE COMPOUND USING 5-METHYLURIDINE AS STARTING RAW MATERIAL. WO2009125841.
  8. METHOD FOR PURIFYING ETHYNYLTHYMIDINE COMPOUND. WO2009119785.
  9. METHOD FOR SYNTHESIZING L-ANSERINE. JP2005082571.
  10. NOVEL 2,4-DIAMINO-1,3,5-TRIAZINE DERIVATIVE. WO2004054989.